What is AM-2233 ?
AM-2233
AM-2233 is a drug that acts as a highly potent full agonist for the cannabinoid receptors, with a Ki of 1.8 nM at CB1 and 2.2 nM at CB2 as the active (R) enantiomer.
It was developed as a selective radioligand for the cannabinoid receptors and has been used as its 131I derivative for mapping the distribution of the CB1 receptor in the brain.
AM-2233 was found to fully substitute for THC in rats, with a potency lower than that of JWH-018 but higher than WIN 55,212-2.
It is notable for inducing tinnitus,though the reasons for this are unclear and may provide valuable insight into tinnitus research.
We are offering am-2233 . Very good product.has very high efficacy.just.production staff are the first to be involved
in quality, since they are made aware that their role is fundamental to reach the goals strativa wants to achieve.in order to guarantee the quality standards of the manufacturing cycle and, consequently,
the quality of its drugs, besides quality control and quality assurance, which are the functions traditionally involved,
strativa has involved in the quality process also the company structures that support production, such as engineering and planning, and obviously all the staff of the plants
Synonym: AM-2233; AM 2233; AM2233; CHEMBL364266;
IUPAC/Chemical Name: 1-((N-Methylpiperidin-2-yl)methyl)-3-(2-iodobenzoyl)indole
InChi Key: KSLCYQTUSSEGPT-UHFFFAOYSA-N
InChi Code: InChI=1S/C22H23IN2O/c1-24-13-7-6-8-16(24)14-25-15-19(17-9-3-5-12-21(17)25)22(26)18-10-2-4-11-20(18)23/h2-5,9-12,15-16H,6-8,13-14H2,1H3
SMILES Code: CN1CCCCC1Cn2cc(C(=O)c3ccccc3I)c4ccccc24
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable
enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).
